Molekulární biofyzika a farmakologie

Novohradsky V., Markova L., Kostrhunova H., Kasparkova J., Hoeschele J., Brabec V. (2022), A [Pt(cis-1,3-diaminocycloalkane)Cl2] analog exhibits hallmarks typical of immunogenic cell death inducers in model cancer cells., Journal of Inorganic Biochemistry

Malina J., Kostrhunova H., Brabec V. (2022), Dinuclear nickel(II) supramolecular helicates down-regulate gene expression in human cells by stabilizing DNA G-quadruplexes formed in the promoter regions, Inorganic Chemistry Frontiers

Markova L., Novohradsky V., Kasparkova J., Ruiz J., Brabec V. (2022), Dipyridophenazine iridium(III) complex as a phototoxic cancer stem cell selective, mitochondria targeting agent, Chemico-Biological Interactions

Hreusova M., Novohradsky V., Markova L., Kostrhunova H., Potočňák I., Brabec V., Kasparkova J. (2022), Gallium(III) complex with cloxyquin ligands induces ferroptosis in cancer cells and is a potent agent against both differentiated and tumorigenic cancer stem Rhabdomyosarcoma cells, Bioinorganic Chemistry and Applications

Kasparkova J., Kostrhunova H., Novohradsky V., Ma L., Zhu G., Milaeva E. R., Shtill A. A., Vinck R., Gasser G., Brabec V., Nazarov A. A. (2022), Is antitumor Pt(IV) complex containing two axial lonidamine ligands a true dual- or multi-action prodrug?, Metallomics

Malina J., Kostrhunova H., Novohradsky V., Scott P., Brabec V. (2022), Metallohelix vectors for efficient gene delivery via cationic DNA nanoparticles., Nucleic Acids Research

Kasparkova J., Kostrhunova H., Novohradsky V., Logvinov A. A., Temnov V. V., Borisova N. E., Podrugina T. A., Markova L., Starha P., Nazarov A. A., Brabec V. (2022), Novel cis-Pt(II) complexes with alkylpyrazole ligands: Synthesis, characterization, and unusual mode of anticancer action, Bioinorganic Chemistry and Applications

Novohradsky V., Markova L., Kostrhunova H., Svitelova M., Kasparkova J., Barbanente A., Papadia P., Margiotta N., Hoeschele J. D., Brabec V. (2022), Pt(II) complex containing the 1R,2R enantiomer of trans-1,2-diamino-4-cyclohexene ligand effectively and selectively inhibits the viability of aggressive pancreatic adenocarcinoma cells and alters their lipid metabolism, Inorganic Chemistry Frontiers

Cervinka J., Gobbo A., Biancalana L., Markova L., Novohradsky V., Guelfi M., Zacchini S., Kasparkova J., Brabec V., Marchetti F. (2022), Ruthenium(II)–tris-pyrazolylmethane complexes inhibit cancer cell growth by disrupting mitochondrial calcium homeostasis, Journal of Medicinal Chemistry